Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50049074
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234032BDBM50234032(CHEMBL4060668)
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234031BDBM50234031(CHEMBL4082542)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234025BDBM50234025(CHEMBL4093791)
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234035BDBM50234035(CHEMBL4070008)
Affinity DataIC50: 450nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234037BDBM50234037(CHEMBL4083510)
Affinity DataIC50: 560nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234024BDBM50234024(CHEMBL4097198)
Affinity DataIC50: 700nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234033BDBM50234033(CHEMBL4078213)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234022BDBM50234022(CHEMBL4066295)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234020BDBM50234020(CHEMBL4101592)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234030BDBM50234030(CHEMBL4101510)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234021BDBM50234021(CHEMBL4074903)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234027BDBM50234027(CHEMBL4086033)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234028BDBM50234028(CHEMBL4063448)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234034BDBM50234034(CHEMBL4093860)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234036BDBM50234036(CHEMBL4064507)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234026BDBM50234026(CHEMBL4073089)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234029BDBM50234029(CHEMBL4091303)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Merck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234019BDBM50234019(CHEMBL4096268)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2019
Entry Details Article
PubMed