Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50048058
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203153(CHEMBL3927163)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203153(CHEMBL3927163)
Affinity DataIC50: 40nMAssay Description:Displacement of [1,2,6,7-3H]-PG from recombinant human GST-tagged PR-LBD (657 to 933 residues) expressed in baculovirus infected insect cells measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203179(CHEMBL3917144)
Affinity DataIC50: 47nMAssay Description:Displacement of [1,2,6,7-3H]-PG from recombinant human GST-tagged PR-LBD (657 to 933 residues) expressed in baculovirus infected insect cells measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203158(CHEMBL3912293)
Affinity DataIC50: 62nMAssay Description:Displacement of [1,2,6,7-3H]-PG from recombinant human GST-tagged PR-LBD (657 to 933 residues) expressed in baculovirus infected insect cells measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203195(CHEMBL3942784)
Affinity DataIC50: 110nMAssay Description:Displacement of [1,2,6,7-3H]-PG from recombinant human GST-tagged PR-LBD (657 to 933 residues) expressed in baculovirus infected insect cells measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203179(CHEMBL3917144)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203170(CHEMBL3936121)
Affinity DataIC50: 140nMAssay Description:Displacement of [1,2,6,7-3H]-PG from recombinant human GST-tagged PR-LBD (657 to 933 residues) expressed in baculovirus infected insect cells measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203170(CHEMBL3936121)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203158(CHEMBL3912293)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203171(CHEMBL3893240)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203180(CHEMBL3945051)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203189(CHEMBL3902219)
Affinity DataIC50: 250nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203222(CHEMBL3911233)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203174(CHEMBL3908173)
Affinity DataIC50: 300nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203180(CHEMBL3945051)
Affinity DataIC50: 310nMAssay Description:Displacement of [1,2,6,7-3H]-PG from recombinant human GST-tagged PR-LBD (657 to 933 residues) expressed in baculovirus infected insect cells measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203154(CHEMBL3953780)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203195(CHEMBL3942784)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203178(CHEMBL3930183)
Affinity DataIC50: 370nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203184(CHEMBL3980435)
Affinity DataIC50: 390nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203212(CHEMBL3895538)
Affinity DataIC50: 410nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203220(CHEMBL3952612)
Affinity DataIC50: 450nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203182(CHEMBL3971739)
Affinity DataIC50: 470nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203176(CHEMBL3986969)
Affinity DataIC50: 490nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203221(CHEMBL3929091)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203187(CHEMBL3915906)
Affinity DataIC50: 510nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203193(CHEMBL3898358)
Affinity DataIC50: 520nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203177(CHEMBL3966839)
Affinity DataIC50: 640nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203183(CHEMBL3903419)
Affinity DataIC50: 650nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203190(CHEMBL3939189)
Affinity DataIC50: 670nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203191(CHEMBL3982227)
Affinity DataIC50: 740nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203185(CHEMBL3961285)
Affinity DataIC50: 810nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203186(CHEMBL3924894)
Affinity DataIC50: 820nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203219(CHEMBL3912431)
Affinity DataIC50: 960nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203218(CHEMBL3930349)
Affinity DataIC50: 990nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203156(CHEMBL3972388)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203157(CHEMBL3943861)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203173(CHEMBL3956621)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203192(CHEMBL3942112)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203217(CHEMBL3926140)
Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203214(CHEMBL3921236)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203159(CHEMBL3970606)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203213(CHEMBL3951528)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203216(CHEMBL3931396)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203223(CHEMBL3983391)
Affinity DataIC50: 2.20E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203215(CHEMBL3949203)
Affinity DataIC50: 2.60E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442126(CHEMBL2441096)
Affinity DataIC50: 2.80E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203155(CHEMBL3940435)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203181(CHEMBL3957844)
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50203172(CHEMBL3917444)
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50442124(CHEMBL2441094)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells incubated for 24 hrs in presence of P4 by alkaline phosphatase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2018
Entry Details Article
PubMed
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