Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50047983
TargetAndrogen receptor(Human)
Chinese Academy of Medical Science

Curated by ChEMBL
LigandPNGBDBM50199857(TRIPTOPHENOLIDE)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at wild type AR in human PC3 cells assessed as suppression of DHT-induced receptor transcriptional activation after 24 hrs by PSA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Chinese Academy of Medical Science

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 294nMAssay Description:Displacement of fluormone-DHT green from His/GST-tagged rat AR ligand binding domain after 4 to 8 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Chinese Academy of Medical Science

Curated by ChEMBL
LigandPNGBDBM50199857(TRIPTOPHENOLIDE)
Affinity DataIC50: 467nMAssay Description:Displacement of fluormone-DHT green from His/GST-tagged rat AR ligand binding domain after 4 to 8 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed