Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50011726
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550378(CHEMBL4799175)
Affinity DataIC50: 140nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550361(CHEMBL4793070)
Affinity DataIC50: 260nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550377(CHEMBL4758277)
Affinity DataIC50: 290nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50135912(5,5-dimethyl-3-[4-nitro-3-(trifluoromethyl)phenyl]...)
Affinity DataIC50: 600nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550354(CHEMBL4787997)
Affinity DataIC50: 910nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550357(CHEMBL4755665)
Affinity DataIC50: 990nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550366(CHEMBL4778298)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550379(CHEMBL4778974)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550372(CHEMBL4750103)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550353(CHEMBL4790269)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550376(CHEMBL4786505)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550350(CHEMBL4786811)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550347(CHEMBL4572306)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550355(CHEMBL4778185)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550370(CHEMBL4799429)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550368(CHEMBL4782426)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550356(CHEMBL4747499)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550362(CHEMBL4743529)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550374(CHEMBL4748557)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550380(CHEMBL4465426)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550367(CHEMBL4748422)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550358(CHEMBL4793158)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550359(CHEMBL4763136)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550373(CHEMBL4781708)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550375(CHEMBL4740944)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550348(CHEMBL4777133)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550351(CHEMBL4777511)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550369(CHEMBL4746443)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550365(CHEMBL4763876)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550364(CHEMBL4743225)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550363(CHEMBL4756377)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550371(CHEMBL4747544)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550360(CHEMBL4782196)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550352(CHEMBL4754845)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50550349(CHEMBL4795534)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of wild-type androgen receptor in human LAPC4 cells assessed as inhibition of DHT-induced luciferase activity measured after 24 hrs by luc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed