Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50048165
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206892(CHEMBL3948489)
Affinity DataIC50: 730nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206895(CHEMBL3983017)
Affinity DataIC50: 830nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206890(CHEMBL3910830)
Affinity DataIC50: 980nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206891(CHEMBL3921785)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206897(CHEMBL3945423)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206885(CHEMBL3930722)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206896(CHEMBL3958208)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206889(CHEMBL3928840)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206893(CHEMBL3901794)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206886(CHEMBL3955393)
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206894(CHEMBL3972865)
Affinity DataIC50: 2.27E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206887(CHEMBL3976003)
Affinity DataIC50: 3.18E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50206888(CHEMBL3984034)
Affinity DataIC50: 3.22E+3nMAssay Description:Inhibition of acetylcholinesterase (unknown origin) assessed as reduction in formation of 5-thio-2-nitrobenzoate from acetylthiocholine iodide preinc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2018
Entry Details Article
PubMed