Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50049112
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234631(CHEMBL4078686)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234634(CHEMBL4100259)
Affinity DataIC50: 17nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234638(CHEMBL4092511)
Affinity DataIC50: 22nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50069985({1-[(S)-(S)-1-((S)-1-Formyl-3-methyl-butylcarbamoy...)
Affinity DataIC50: 25nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234630(CHEMBL4077762)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234655(CHEMBL4102028)
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234653(CHEMBL4066773)
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234641(CHEMBL4093360)
Affinity DataIC50: 3.57E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234654(CHEMBL4072644)
Affinity DataIC50: 5.84E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234636(CHEMBL4083790)
Affinity DataIC50: 8.83E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234634(CHEMBL4100259)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using (Z)-LLE-bNA as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234635(CHEMBL4073408)
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234659(CHEMBL4062055)
Affinity DataIC50: 2.22E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234639(CHEMBL4064046)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234636(CHEMBL4083790)
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using (Z)-LLE-bNA as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234638(CHEMBL4092511)
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using (Z)-LLE-bNA as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234642(CHEMBL4094297)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-1(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234631(CHEMBL4078686)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using (Z)-LLE-bNA as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234640(CHEMBL4085613)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234637(CHEMBL4070680)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234633(CHEMBL4064812)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-2(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234638(CHEMBL4092511)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Bz-VGR-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234632(CHEMBL4096708)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2019
Entry Details Article
PubMed