Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 7890
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223126(P5i-7)
Affinity DataIC50: 720nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223131(2-((5-(4-methoxyphenyl)furan-2-yl)methylene)hydraz...)
Affinity DataIC50: 2.10E+3nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223136(2-((6-(4-chlorophenyl)pyridin-2-yl)methylene)hydra...)
Affinity DataIC50: 3.50E+3nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223134(2-((4′-chloro-[1,1′-biphenyl]-3-yl)met...)
Affinity DataIC50: 3.80E+3nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223135(2-((5-(4-chlorophenyl)pyridin-3-yl)methylene)hydra...)
Affinity DataIC50: 6.90E+3nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223127(2-((5-phenylfuran-2-yl)methylene)hydrazinecarboxam...)
Affinity DataIC50: 1.20E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223129(2-((5-(4-fluorophenyl)furan-2-yl)methylene)hydrazi...)
Affinity DataIC50: 1.20E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223133(2-((5-(2-amino-4-chlorophenyl)furan-2-yl)methylene...)
Affinity DataIC50: 1.30E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223128(2-((5-(3-fluorophenyl)furan-2-yl)methylene)hydrazi...)
Affinity DataIC50: 1.40E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223130(2-((5-(4-nitrophenyl)furan-2-yl)methylene)hydrazin...)
Affinity DataIC50: 1.80E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM223132(2-((5-(4-aminophenyl)furan-2-yl)methylene)hydrazin...)
Affinity DataIC50: 4.00E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Sichuan University

LigandPNGBDBM8460(5-{[5-(4-chlorophenyl)furan-2-yl]methylidene}-2-su...)
Affinity DataIC50: 6.70E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3 [N508S](Human)
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 6(Human)
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 8(Human)
Sichuan University

LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed