Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50048269
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210860(CHEMBL3936390)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210866(CHEMBL3979767)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210858(CHEMBL3906952)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50243008(N,N-Diethyl-2-(2-(4-(3-fluoropropoxy)phenyl)-5,7-d...)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50243007(N,N-diethyl-2-(2-(4-(2-fluoroethoxy)phenyl)-5,7-di...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210857(CHEMBL3938340)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210864(CHEMBL3960249)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210867(CHEMBL3923539)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210863(CHEMBL3929294)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210859(CHEMBL3908452)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210865(CHEMBL3909555)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210861(CHEMBL3896806)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210868(CHEMBL3981447)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210856(CHEMBL3906707)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Institute of Biomedical Imaging (I2Bm)

Curated by ChEMBL
LigandPNGBDBM50210862(CHEMBL3920384)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2018
Entry Details Article
PubMed