Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50047954
TargetProtein polybromo-1(Human)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50198438(CHEMBL3904183)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to N-terminal his6-tagged human PB1 bromodomain 5 expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 at 15 uM by ITC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProtein polybromo-1(Human)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50198451(CHEMBL1491707)
Affinity DataKd:  3.40E+3nMAssay Description:Binding affinity to N-terminal his6-tagged human PB1 bromodomain 5 expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 at 15 uM by ITC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProtein polybromo-1(Human)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50198448(CHEMBL3966713)
Affinity DataKd:  3.40E+3nMAssay Description:Binding affinity to N-terminal his6-tagged human PB1 bromodomain 5 expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 at 15 uM by ITC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProtein polybromo-1(Human)
University of Athens

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataKd:  1.29E+4nMAssay Description:Binding affinity to N-terminal his6-tagged human PB1 bromodomain 5 expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 at 15 uM by ITC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein polybromo-1(Human)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50198440(CHEMBL3945847)
Affinity DataKd:  1.15E+4nMAssay Description:Binding affinity to N-terminal his6-tagged human PB1 bromodomain 5 expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 at 15 uM by ITC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProtein polybromo-1(Human)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50198447(CHEMBL3899245)
Affinity DataKd:  43nMAssay Description:Binding affinity to N-terminal his6-tagged human PB1 bromodomain 5 expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 at 15 uM by ITC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProtein polybromo-1(Human)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50198450(CHEMBL3927964)
Affinity DataKd:  5.10E+3nMAssay Description:Binding affinity to N-terminal his6-tagged human PB1 bromodomain 5 expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 at 15 uM by ITC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed
TargetProtein polybromo-1(Human)
University of Athens

Curated by ChEMBL
LigandPNGBDBM50198449(CHEMBL3936967)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to N-terminal his6-tagged human PB1 bromodomain 5 expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 at 15 uM by ITC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2018
Entry Details Article
PubMed