Compile Data Set for Download or QSAR
Report error Found 202 Enz. Inhib. hit(s) with all data for entry = 50009973
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533873(CHEMBL4585638)
Affinity DataIC50: 0.140nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533953(CHEMBL4474379)
Affinity DataIC50: 0.160nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533933(CHEMBL4566719)
Affinity DataIC50: 0.170nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533944(CHEMBL4516712)
Affinity DataIC50: 0.170nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533855(CHEMBL4582367)
Affinity DataIC50: 0.230nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533865(CHEMBL4539811)
Affinity DataIC50: 0.310nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533904(CHEMBL4447139)
Affinity DataIC50: 0.320nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533862(CHEMBL4544693)
Affinity DataIC50: 0.330nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533897(CHEMBL4474058)
Affinity DataIC50: 0.380nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533901(CHEMBL4460880)
Affinity DataIC50: 0.390nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533938(CHEMBL4449450)
Affinity DataIC50: 0.390nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533976(CHEMBL4526641)
Affinity DataIC50: 0.390nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533911(CHEMBL4443108)
Affinity DataIC50: 0.410nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533858(CHEMBL4449332)
Affinity DataIC50: 0.440nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533903(CHEMBL4436854)
Affinity DataIC50: 0.450nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533863(CHEMBL4593521)
Affinity DataIC50: 0.580nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50162007(3-[(2R)-amino-2-phenylethyl]-1-(2,6-difluorobenzyl...)
Affinity DataIC50: 0.590nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533948(CHEMBL4446435)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533943(CHEMBL4540232)
Affinity DataIC50: 0.680nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533858(CHEMBL4449332)
Affinity DataIC50: 0.760nMAssay Description:Antagonist activity against human GnRH receptor expressed in human Chem1 cells assessed as inhibition of LHRH-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533863(CHEMBL4593521)
Affinity DataIC50: 0.860nMAssay Description:Antagonist activity against human GnRH receptor expressed in human Chem1 cells assessed as inhibition of LHRH-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533955(CHEMBL4563562)
Affinity DataIC50: 0.910nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533945(CHEMBL4463476)
Affinity DataIC50: 0.950nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533902(CHEMBL4446131)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533912(CHEMBL4576169)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533877(CHEMBL4563686)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533892(CHEMBL4456703)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533967(CHEMBL4452347)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533932(CHEMBL4522657)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533859(CHEMBL4464132)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533864(CHEMBL4550720)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533876(CHEMBL4461692)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533946(CHEMBL4474116)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533934(CHEMBL4467407)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533917(CHEMBL4556717)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533863(CHEMBL4593521)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity against human GnRH receptor expressed in HEK293 cells co-transfected with pGL4-NFAT promoter AP1-luc assessed as inhibition of 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533868(CHEMBL4557575)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533874(CHEMBL4590493)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533891(CHEMBL4467261)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533900(CHEMBL4456937)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533893(CHEMBL4583933)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533890(CHEMBL4567165)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533875(CHEMBL4585969)
Affinity DataIC50: 2.80nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533858(CHEMBL4449332)
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity against human GnRH receptor expressed in HEK293 cells assessed as reduction in ERK1/2 phosphorylation pre-incubated for 5 mins be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50291832(CHEMBL4173938)
Affinity DataIC50: 2.90nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533918(CHEMBL4515452)
Affinity DataIC50: 3.10nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rhesus macaque)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533863(CHEMBL4593521)
Affinity DataIC50: 3.5nMAssay Description:Displacement of [125I]D-Trp6-LHRH from monkey GnRH receptor expressed in HEK293 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rhesus macaque)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533858(CHEMBL4449332)
Affinity DataIC50: 3.70nMAssay Description:Displacement of [125I]D-Trp6-LHRH from monkey GnRH receptor expressed in HEK293 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533878(CHEMBL4517137)
Affinity DataIC50: 3.80nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Sk Chemicals

Curated by ChEMBL
LigandPNGBDBM50533920(CHEMBL4451280)
Affinity DataIC50: 3.80nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cell membranes incubated for 1 hr by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
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