Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50010254
TargetBromodomain-containing protein 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM209487(US9266891, III-28 | US10328074, Example III-28 | U...)
Affinity DataIC50: 1nMAssay Description:Displacement of biotinylated tetra-acetylated histone H4 peptide from GST-tagged BRD4-BD1 (44 to 168 residues) (unknown origin) measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM209485(US9266891, III-26 | US10328074, Example III-26 | U...)
Affinity DataIC50: 5nMAssay Description:Displacement of biotinylated tetra-acetylated histone H4 peptide from GST-tagged BRD4-BD1 (44 to 168 residues) (unknown origin) measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM209453(US9266891, I-5 | US10328074, Example I-5 | US11077...)
Affinity DataIC50: 8nMAssay Description:Displacement of biotinylated tetra-acetylated histone H4 peptide from GST-tagged BRD4-BD1 (44 to 168 residues) (unknown origin) measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM209472(US9266891, III-13 | US10328074, Example III-13 | U...)
Affinity DataIC50: 9nMAssay Description:Displacement of biotinylated tetra-acetylated histone H4 peptide from GST-tagged BRD4-BD1 (44 to 168 residues) (unknown origin) measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM209458(US9266891, II-2 | US10328074, Example II-2 | US110...)
Affinity DataIC50: 15nMAssay Description:Displacement of biotinylated tetra-acetylated histone H4 peptide from GST-tagged BRD4-BD1 (44 to 168 residues) (unknown origin) measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM209498(US9266891, III-39 | US10328074, Example III-39 | U...)
Affinity DataIC50: 126nMAssay Description:Displacement of biotinylated tetra-acetylated histone H4 peptide from GST-tagged BRD4-BD1 (44 to 168 residues) (unknown origin) measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed