Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50010054
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534765(CHEMBL4443952)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534753(CHEMBL4578460)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534766(CHEMBL4539641)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534752(CHEMBL4552325)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534764(CHEMBL4476854)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534760(CHEMBL4582423)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534749(CHEMBL4437901)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534761(CHEMBL4467949)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534754(CHEMBL4458142)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534750(CHEMBL4461741)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534756(CHEMBL4468577)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534758(CHEMBL4473908)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534762(CHEMBL4589258)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534755(CHEMBL4528003)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534757(CHEMBL4455924)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534768(CHEMBL4583172)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534767(CHEMBL4542515)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534759(CHEMBL4571149)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataIC50: 11nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534763(CHEMBL4514997)
Affinity DataIC50: 14nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50248088(N-(4-(2-(1-ethyl-1H-imidazol-4-yl)thieno[3,2-b]pyr...)
Affinity DataIC50: 29nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM24485(3-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophe...)
Affinity DataIC50: 80nMAssay Description:Inhibition of c-Met (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534751(CHEMBL4527370)
Affinity DataIC50: 105nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50534748(CHEMBL4461009)
Affinity DataIC50: 133nMAssay Description:Inhibition of recombinant c-Met (unknown origin) using poly (Glu,Tyr)4:1 as substrate incubated for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed