Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50047748
TargetType-1 angiotensin II receptor(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 3.20nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50187505(CHEMBL1332729)
Affinity DataIC50: 199nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50187505(CHEMBL1332729)
Affinity DataIC50: 200nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50187507(CHEMBL1374011)
Affinity DataIC50: 2.09E+3nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50187509(CHEMBL1474431)
Affinity DataIC50: 2.19E+3nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50187506(CHEMBL1716544)
Affinity DataIC50: 2.57E+3nMAssay Description:Displacement of [125I-Sar1-Ile8]Ang2 from human AT1 receptor expressed in HEK293 cell membrane incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed