Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50048144
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM13216(N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyeth...)
Affinity DataIC50: 4nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206297(CHEMBL3911525)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant human Src using KVEKIGEGTYGVVYK as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206301(CHEMBL3954137)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206297(CHEMBL3911525)
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206296(CHEMBL3904850)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of recombinant human Src using KVEKIGEGTYGVVYK as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206296(CHEMBL3904850)
Affinity DataIC50: 2.61E+4nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206298(CHEMBL3917521)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206300(CHEMBL3967164)
Affinity DataIC50: 6.56E+4nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206301(CHEMBL3954137)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of recombinant human Src using KVEKIGEGTYGVVYK as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206302(CHEMBL3983676)
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50206299(CHEMBL3908573)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of wild type recombinant human Abl using abtide as substrate by [gamma-32P]ATP based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Cairo University

Curated by ChEMBL
LigandPNGBDBM50354485(CHEMBL412298)
Affinity DataKi:  40nMAssay Description:Inhibition of wild type Abl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2018
Entry Details Article
PubMed