Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 7533
TargetAdenosine receptor A1(Human)
Uppsala University

LigandPNGBDBM50060165(1-DEAZA-ADENOSINE | (2R,3R,4S,5R)-2-(7-Amino-imida...)
Affinity DataKi:  84nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

LigandPNGBDBM200215(Adenosine receptor agonist, 11)
Affinity DataKi:  130nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

LigandPNGBDBM200213(Adenosine receptor agonist, 9)
Affinity DataKi:  348nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

LigandPNGBDBM200217(Adenosine receptor agonist, 14)
Affinity DataKi:  359nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

LigandPNGBDBM82055(CAS_6736-58-9 | 3-DEAZAADENOSINE | 9-Deazaado | Ad...)
Affinity DataKi:  461nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

LigandPNGBDBM200213(Adenosine receptor agonist, 9)
Affinity DataKi:  467nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

LigandPNGBDBM200213(Adenosine receptor agonist, 9)
Affinity DataKi:  495nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

LigandPNGBDBM200217(Adenosine receptor agonist, 14)
Affinity DataKi:  557nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

LigandPNGBDBM50060165(1-DEAZA-ADENOSINE | (2R,3R,4S,5R)-2-(7-Amino-imida...)
Affinity DataKi:  583nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Uppsala University

LigandPNGBDBM50060165(1-DEAZA-ADENOSINE | (2R,3R,4S,5R)-2-(7-Amino-imida...)
Affinity DataKi:  645nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

LigandPNGBDBM200211(Adenosine receptor agonist, 7)
Affinity DataKi:  823nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

LigandPNGBDBM200215(Adenosine receptor agonist, 11)
Affinity DataKi:  917nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

LigandPNGBDBM50424715(Ladakamycin | Vidaza | U-18496 | AZACITIDINE | Ade...)
Affinity DataKi:  2.01E+3nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

LigandPNGBDBM50424715(Ladakamycin | Vidaza | U-18496 | AZACITIDINE | Ade...)
Affinity DataKi:  3.68E+3nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Uppsala University

LigandPNGBDBM50154375(Tribavirin | cid_37542 | Ribavirin | Adenosine rec...)
Affinity DataKi:  7.41E+3nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Uppsala University

LigandPNGBDBM200216(Adenosine receptor agonist, 13)
Affinity DataKi:  8.02E+3nMAssay Description:Radioligand binding assays were performed using membranes prepared from CHO (hA1AR or hA3AR) or HEK293 (hA2AAR) cells stably expressing a single hAR ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details Article
PubMed