Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50001807
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50002022(CHEMBL16779 | (2-Benzyl-3-hydroxycarbamoyl-propion...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018211(CHEMBL36094 | 3-(2-Benzyl-3-hydroxycarbamoyl-propi...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018211(CHEMBL36094 | 3-(2-Benzyl-3-hydroxycarbamoyl-propi...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018216(CHEMBL290337 | 2-Benzyl-3-(2-benzyl-3-hydroxycarba...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018220(CHEMBL37921 | 3-(2-Benzyl-3-hydroxycarbamoyl-propi...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018212(CHEMBL440104 | 3-(2-Benzyl-3-hydroxycarbamoyl-prop...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018218(CHEMBL37418 | (R,S)2-(2-Benzyl-3-hydroxycarbamoyl-...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50405952(CHEMBL2114407)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50405951(CHEMBL2115347)
Affinity DataIC50: 3nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50405949(CHEMBL2114408)
Affinity DataIC50: 3nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50405950(CHEMBL2115348)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018213(CHEMBL285617 | 3-(2-Benzyl-3-hydroxycarbamoyl-prop...)
Affinity DataIC50: 13nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018213(CHEMBL285617 | 3-(2-Benzyl-3-hydroxycarbamoyl-prop...)
Affinity DataIC50: 13nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50405949(CHEMBL2114408)
Affinity DataIC50: 23nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018214(CHEMBL417878 | 4-(2-Benzyl-3-hydroxycarbamoyl-prop...)
Affinity DataIC50: 28nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50405952(CHEMBL2114407)
Affinity DataIC50: 33nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018217(CHEMBL36841 | 5-(2-Benzyl-3-hydroxycarbamoyl-propi...)
Affinity DataIC50: 52nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018216(CHEMBL290337 | 2-Benzyl-3-(2-benzyl-3-hydroxycarba...)
Affinity DataIC50: 72nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018219(CHEMBL290366 | 2-[(2-Benzyl-3-hydroxycarbamoyl-pro...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018218(CHEMBL37418 | (R,S)2-(2-Benzyl-3-hydroxycarbamoyl-...)
Affinity DataIC50: 130nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Rabbit)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018219(CHEMBL290366 | 2-[(2-Benzyl-3-hydroxycarbamoyl-pro...)
Affinity DataIC50: 150nMAssay Description:Inhibition of neutral endopeptidase activity in rabbit kidney with 20 nM [3H]D-Ala2-Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018211(CHEMBL36094 | 3-(2-Benzyl-3-hydroxycarbamoyl-propi...)
Affinity DataIC50: 350nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018211(CHEMBL36094 | 3-(2-Benzyl-3-hydroxycarbamoyl-propi...)
Affinity DataIC50: 350nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018220(CHEMBL37921 | 3-(2-Benzyl-3-hydroxycarbamoyl-propi...)
Affinity DataIC50: 360nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50405951(CHEMBL2115347)
Affinity DataIC50: 400nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018217(CHEMBL36841 | 5-(2-Benzyl-3-hydroxycarbamoyl-propi...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018212(CHEMBL440104 | 3-(2-Benzyl-3-hydroxycarbamoyl-prop...)
Affinity DataIC50: 670nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50405950(CHEMBL2115348)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50018214(CHEMBL417878 | 4-(2-Benzyl-3-hydroxycarbamoyl-prop...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50002022(CHEMBL16779 | (2-Benzyl-3-hydroxycarbamoyl-propion...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Aminopeptidase N activity in pig kidney with 10 nM [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed