Compile Data Set for Download or QSAR
Report error Found 140 Enz. Inhib. hit(s) with all data for entry = 50009846
TargetSTE20-like serine/threonine-protein kinase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  240nMAssay Description:Binding affinity to human SLKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532786(CHEMBL4513513)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to human AXL by active site dependent completion binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  4nMAssay Description:Binding affinity to human FLT3More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human ALKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  50nMAssay Description:Binding affinity to human TRKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor TYRO3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  58nMAssay Description:Binding affinity to human Tyro3More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  50nMAssay Description:Binding affinity to human TRKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  38nMAssay Description:Binding affinity to human MEK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  10nMAssay Description:Binding affinity to human LOKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  11nMAssay Description:Binding affinity to human HIPk4More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  4nMAssay Description:Binding affinity to human FLT3More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCyclin-dependent kinase 11B(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  470nMAssay Description:Binding affinity to human CDK11More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  200nMAssay Description:Binding affinity to human BLKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human ALKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  2.70nMAssay Description:Binding affinity to human AXL by active site dependent completion binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBDNF/NT-3 growth factors receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  54nMAssay Description:Binding affinity to human TRKBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetSTE20-like serine/threonine-protein kinase(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  240nMAssay Description:Binding affinity to human SLKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  1.40nMAssay Description:Binding affinity to human MERMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 5(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  38nMAssay Description:Binding affinity to human MEK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  10nMAssay Description:Binding affinity to human LOKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCyclin-dependent kinase 11B(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  470nMAssay Description:Binding affinity to human CDK11More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  200nMAssay Description:Binding affinity to human BLKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  2.70nMAssay Description:Binding affinity to human AXL by active site dependent completion binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532786(CHEMBL4513513)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to human AXL by active site dependent completion binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  79nMAssay Description:Binding affinity to human METMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  1.67E+3nMAssay Description:Binding affinity to human KITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  2.70nMAssay Description:Binding affinity to human AXLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  1.40nMAssay Description:Binding affinity to human MERMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetBDNF/NT-3 growth factors receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  54nMAssay Description:Binding affinity to human TRKBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor TYRO3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  58nMAssay Description:Binding affinity to human Tyro3More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human CDK8More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  79nMAssay Description:Binding affinity to human METMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  11nMAssay Description:Binding affinity to human HIPk4More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  2.70nMAssay Description:Binding affinity to human AXLMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCyclin-dependent kinase 8(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human CDK8More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataKd:  1.67E+3nMAssay Description:Binding affinity to human KITMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50172079(CHEMBL3809489 | US20250026773, Positive Drug 1 BGB...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50172079(CHEMBL3809489 | US20250026773, Positive Drug 1 BGB...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532786(CHEMBL4513513)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532786(CHEMBL4513513)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant AXL incubated for 1 to 1.5 hrs by FRET based Z'-Lyte kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50172077(CHEMBL3810063)
Affinity DataIC50: 10nMAssay Description:Inhibition of Axl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataIC50: 10nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50172077(CHEMBL3810063)
Affinity DataIC50: 10nMAssay Description:Inhibition of Axl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50532781(CHEMBL4571241)
Affinity DataIC50: 10nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50172079(CHEMBL3809489 | US20250026773, Positive Drug 1 BGB...)
Affinity DataIC50: 14nMAssay Description:Inhibition of Axl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50172079(CHEMBL3809489 | US20250026773, Positive Drug 1 BGB...)
Affinity DataIC50: 14nMAssay Description:Inhibition of Axl (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
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