Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50010011
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)
Affinity DataKd:  169nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50534392(CHEMBL4446324)
Affinity DataKd:  2.56E+4nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHeat shock protein 90, putative(Plasmodium falciparum (isolate 3D7))
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50406805(CHEMBL585793 | GNF-Pf-4574)
Affinity DataKd:  2.81E+4nMAssay Description:Binding affinity to recombinant Plasmodium falciparum Hsp90 expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-beta(Human)
University of Geneva

Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)
Affinity DataKd:  158nMAssay Description:Binding affinity to recombinant human Hsp90 beta expressed in Escherichia coli BL21(DE3) pLysS by microscale thermophoresis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed