Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50047725
TargetMu-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185754(CHEMBL3822676)
Affinity DataIC50: 14nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185755(CHEMBL3823054)
Affinity DataIC50: 18nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataIC50: 23nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185752(CHEMBL3822822)
Affinity DataIC50: 56nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185754(CHEMBL3822676)
Affinity DataIC50: 137nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50016867((S)-6-Amino-2-((S)-2-{(R)-2-[(S)-2-amino-3-(4-hydr...)
Affinity DataIC50: 254nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185755(CHEMBL3823054)
Affinity DataIC50: 290nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185753(CHEMBL3822702)
Affinity DataIC50: 410nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185752(CHEMBL3822822)
Affinity DataIC50: 755nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50016867((S)-6-Amino-2-((S)-2-{(R)-2-[(S)-2-amino-3-(4-hydr...)
Affinity DataIC50: 781nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185753(CHEMBL3822702)
Affinity DataIC50: 7.17E+3nMAssay Description:Agonist activity at delta opioid receptor in albino mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataKi:  0.143nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185754(CHEMBL3822676)
Affinity DataKi:  0.367nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185755(CHEMBL3823054)
Affinity DataKi:  0.458nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185752(CHEMBL3822822)
Affinity DataKi:  0.875nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50016867((S)-6-Amino-2-((S)-2-{(R)-2-[(S)-2-amino-3-(4-hydr...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185753(CHEMBL3822702)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185754(CHEMBL3822676)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185752(CHEMBL3822822)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185755(CHEMBL3823054)
Affinity DataKi:  381nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185753(CHEMBL3822702)
Affinity DataKi:  472nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185754(CHEMBL3822676)
Affinity DataKi:  573nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50010483(CHEMBL2181202)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185752(CHEMBL3822822)
Affinity DataKi:  2.36E+3nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185755(CHEMBL3823054)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50016867((S)-6-Amino-2-((S)-2-{(R)-2-[(S)-2-amino-3-(4-hydr...)
Affinity DataKi:  4.23E+3nMAssay Description:Displacement of [3H]U69,593 from kappa-type opioid receptor in guniea pig brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50185753(CHEMBL3822702)
Affinity DataKi:  4.67E+3nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Nanjing Medical University

Curated by ChEMBL
LigandPNGBDBM50016867((S)-6-Amino-2-((S)-2-{(R)-2-[(S)-2-amino-3-(4-hydr...)
Affinity DataKi:  1.92E+4nMAssay Description:Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMed