Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50047615
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178989(CHEMBL3814102)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178987(CHEMBL3814074)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178986(CHEMBL3813832)
Affinity DataIC50: 3.99E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178991(CHEMBL3814875)
Affinity DataIC50: 4.38E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataIC50: 4.43E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178990(CHEMBL2286425)
Affinity DataIC50: 4.57E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50179181(CHEMBL3813799)
Affinity DataIC50: 4.67E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178984(CHEMBL3814404)
Affinity DataIC50: 4.82E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178985(CHEMBL2286727)
Affinity DataIC50: 5.81E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178992(CHEMBL3814906)
Affinity DataIC50: 6.44E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50179088(CHEMBL2286725)
Affinity DataIC50: 7.36E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178983(CHEMBL3814913)
Affinity DataIC50: 7.99E+4nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed
TargetATP-dependent translocase ABCB1(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50178982(CHEMBL2228438)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human P-glycoprotein transfected in pig LLC-GA5-COL150 cells assessed as quinidine transport from apical to basolateral side preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2017
Entry Details Article
PubMed