Compile Data Set for Download or QSAR
Report error Found 87 Enz. Inhib. hit(s) with all data for entry = 50001784
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018100(CHEMBL20721 | (+/-)-trans-2-hydroxy-3-(4-phenylpip...)
Affinity DataIC50: 10nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018100(CHEMBL20721 | (+/-)-trans-2-hydroxy-3-(4-phenylpip...)
Affinity DataIC50: 10nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018108(trans-(4S)-4-tert-butyl-2-(4-phenylpiperidin-1-yl)...)
Affinity DataIC50: 20nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataIC50: 20nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018078(CHEMBL20943 | V-100 | 2-(4-Phenyl-piperidin-1-yl)-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018078(CHEMBL20943 | V-100 | 2-(4-Phenyl-piperidin-1-yl)-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018117(CHEMBL21309 | 2-(4-Cyclohexyl-piperidin-1-yl)-cycl...)
Affinity DataIC50: 40nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018090(CHEMBL20382 | N-[6-Hydroxy-7-(4-phenyl-piperidin-1...)
Affinity DataIC50: 50nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018134(CHEMBL20499 | N-[6-Hydroxy-7-(4-phenyl-piperidin-1...)
Affinity DataIC50: 50nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018127(CHEMBL21271 | 1-[1-(2-Hydroxy-cyclohexyl)-4-phenyl...)
Affinity DataIC50: 50nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018148(CHEMBL21151 | 3-(4-Phenyl-piperidin-1-yl)-1,2,3,4-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018125(CHEMBL21243 | 2-[4-(3-Phenyl-propyl)-piperidin-1-y...)
Affinity DataIC50: 70nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018098(CHEMBL21722 | 5-tert-Butyl-2-(4-phenyl-piperidin-1...)
Affinity DataIC50: 90nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018146(CHEMBL20481 | 2-(4-o-Tolyl-piperazin-1-yl)-cyclohe...)
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018080(CHEMBL20881 | 5-(2-Oxo-hexahydro-thieno[3,4-d]imid...)
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018135(CHEMBL282894 | 2-[4-(4-Nitro-phenyl)-piperidin-1-y...)
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018129(CHEMBL20479 | 3-(4-Phenyl-3,6-dihydro-2H-pyridin-1...)
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018072(CHEMBL278303 | 3-(4-Phenyl-piperidin-1-yl)-cyclohe...)
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018115(CHEMBL281595 | 2-[4-(2,5-Dimethyl-phenyl)-piperazi...)
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018079(CHEMBL277630 | 5-Amino-3-(4-phenyl-piperidin-1-yl)...)
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018110(CHEMBL21165 | 2-[4-(4-Chloro-phenyl)-piperidin-1-y...)
Affinity DataIC50: 100nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018091(CHEMBL278834 | 2-(4-Phenyl-3,6-dihydro-2H-pyridin-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018092(CHEMBL20431 | 1-(2-Hydroxy-cyclohexyl)-4-phenyl-pi...)
Affinity DataIC50: 200nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018071(CHEMBL266183 | 5-(2-Oxo-hexahydro-thieno[3,4-d]imi...)
Affinity DataIC50: 200nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018132(CHEMBL20720 | 2-(4-{3-[1-(2-hydroxycyclohexyl)hexa...)
Affinity DataIC50: 200nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018076(CHEMBL277033 | 2-[4-(4-Chloro-phenyl)-3,6-dihydro-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018147(CHEMBL20429 | N-{4-[1-(2-Hydroxy-cyclohexyl)-piper...)
Affinity DataIC50: 200nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018138(CHEMBL416916 | 8-Amino-3-(4-phenyl-piperidin-1-yl)...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018101(CHEMBL278382 | N-[6-Hydroxy-4-iodo-7-(4-phenyl-pip...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018106(CHEMBL283140 | 1-(4-Phenyl-piperidin-1-yl)-butan-2...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018112(CHEMBL279485 | 2-(4-Benzo[1,3]dioxol-5-ylmethyl-pi...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018085(CHEMBL21152 | (+/-)-trans-2-hydroxy-3-(4-(2-methox...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018082(CHEMBL20719 | 2-(4-Phenyl-piperazin-1-yl)-cyclohex...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018150(CHEMBL21148 | 2-[4-(4-Methoxy-phenyl)-piperazin-1-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018111(CHEMBL20664 | 2-(3-Methyl-4-phenyl-piperazin-1-yl)...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018122(CHEMBL20928 | 2-(4-Benzyl-piperidin-1-yl)-cyclohex...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018104(CHEMBL20689 | 2-[4-(4-Dimethylamino-phenyl)-piperi...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018085(CHEMBL21152 | (+/-)-trans-2-hydroxy-3-(4-(2-methox...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018124(CHEMBL22052 | 2-[4-(2,4-Dinitro-phenyl)-piperidin-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018089(CHEMBL20491 | 2-[4-(4-Methylamino-phenyl)-piperidi...)
Affinity DataIC50: 400nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018086(CHEMBL20744 | 2-[4-(4-Amino-phenyl)-piperidin-1-yl...)
Affinity DataIC50: 500nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018096(CHEMBL20657 | 4-(4-Chloro-phenyl)-1-(2-hydroxy-cyc...)
Affinity DataIC50: 500nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018099(CHEMBL417277 | N-[7-Hydroxy-6-(4-phenyl-piperidin-...)
Affinity DataIC50: 500nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018120(CHEMBL277861 | 2-(4-Phenyl-piperidin-1-yl)-cyclohe...)
Affinity DataIC50: 500nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018130(CHEMBL20593 | 2-Phenyl-6-(4-phenyl-piperidin-1-yl)...)
Affinity DataIC50: 600nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018105(CHEMBL20502 | Acetic acid 1-(4-phenyl-piperidin-1-...)
Affinity DataIC50: 800nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018131(CHEMBL21375 | 4-Hydroxymethyl-2-(4-phenyl-piperidi...)
Affinity DataIC50: 800nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018142(CHEMBL278758 | 1-(2-Hydroxy-cyclohexyl)-1-methyl-4...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50405945(CHEMBL2079585)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50018102(CHEMBL20601 | 1-[1-(2-Hydroxy-cyclohexyl)-piperidi...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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