Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50047606
TargetMonocarboxylate transporter 1(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM214702(US9296728, 25)
Affinity DataIC50: 90nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetMonocarboxylate transporter 1(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM214700(US9296728, 23)
Affinity DataIC50: 170nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetMonocarboxylate transporter 1(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM214701(US9296728, 24)
Affinity DataIC50: 210nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetMonocarboxylate transporter 1(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50442702(CHEMBL2442511 | US9296728, 26)
Affinity DataIC50: 380nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetMonocarboxylate transporter 1(Rat)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM214699(US9296728, 22)
Affinity DataIC50: 450nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed