Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 50047604
LigandPNGBDBM50178285(CHEMBL3813865)
Affinity DataIC50: 13nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM17053(N-(3-{[5-bromo-2-({3-[(pyrrolidin-1-ylcarbonyl)ami...)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant PDK1 assessed as PtdIns-3,4-P2-mediated AKT2 activation using biotin-ARRRDGGGAQPFRPRAATF as substrate after 2 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50178291(CHEMBL3814140)
Affinity DataIC50: 58nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178290(CHEMBL3814770)
Affinity DataIC50: 82nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178293(CHEMBL3815046)
Affinity DataIC50: 84nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178287(CHEMBL3814785)
Affinity DataIC50: 85nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178292(CHEMBL3813933)
Affinity DataIC50: 110nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178284(CHEMBL3814317)
Affinity DataIC50: 120nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178283(CHEMBL3814154)
Affinity DataIC50: 170nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178286(CHEMBL3814539)
Affinity DataIC50: 260nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178277(CHEMBL3814554)
Affinity DataIC50: 390nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178282(CHEMBL3813886)
Affinity DataIC50: 450nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178279(CHEMBL3814704)
Affinity DataIC50: 480nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178281(CHEMBL3814357)
Affinity DataIC50: 500nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178278(CHEMBL3813908)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178298(CHEMBL3799935)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178294(CHEMBL3814340)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178262(CHEMBL3814391)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178263(CHEMBL3814350)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178264(CHEMBL3814929)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178293(CHEMBL3815046)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of PDK1 in human PC3 cells assessed as reduction in AKT Thr308 phosphorylation after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178288(CHEMBL3813849)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178289(CHEMBL3814343)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178280(CHEMBL3813962)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178290(CHEMBL3814770)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178293(CHEMBL3815046)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of PI3K delta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178292(CHEMBL3813933)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178285(CHEMBL3813865)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of PDK1 in human PC3 cells assessed as reduction in AKT Thr308 phosphorylation after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM10838(3-(2-aminopyrimidin-4-yl)-1H-indol-4-ol | Meridian...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human PDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178293(CHEMBL3815046)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50371404(MERIOLIN 1)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human PDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50371404(MERIOLIN 1)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178285(CHEMBL3813865)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50385999(CHEMBL2042885)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human His6-tagged PDK1 using biotinylated PDKtide as substrate after 60 mins by topcount methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178285(CHEMBL3813865)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178292(CHEMBL3813933)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of PDK1 in human PC3 cells assessed as reduction in AKT Thr308 phosphorylation after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178284(CHEMBL3814317)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178294(CHEMBL3814340)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178283(CHEMBL3814154)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178294(CHEMBL3814340)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDK1 in human PC3 cells assessed as reduction in AKT Thr308 phosphorylation after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178286(CHEMBL3814539)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50371404(MERIOLIN 1)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PDK1 in human PC3 cells assessed as reduction in AKT Thr308 phosphorylation after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178294(CHEMBL3814340)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K beta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50371404(MERIOLIN 1)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178284(CHEMBL3814317)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178294(CHEMBL3814340)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178283(CHEMBL3814154)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178290(CHEMBL3814770)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178291(CHEMBL3814140)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
LigandPNGBDBM50178286(CHEMBL3814539)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3K gamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
Displayed 1 to 50 (of 96 total ) | Next | Last >>
Jump to: