Compile Data Set for Download or QSAR
Report error Found 97 Enz. Inhib. hit(s) with all data for entry = 50047499
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171461(CHEMBL3805120)
Affinity DataEC50:  74nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171401(CHEMBL3805860)
Affinity DataEC50:  4.30nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171402(CHEMBL3805099)
Affinity DataEC50:  2.70nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171403(CHEMBL3805704)
Affinity DataEC50:  5.10nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171404(CHEMBL3805649)
Affinity DataEC50:  6nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171405(CHEMBL3805165)
Affinity DataEC50:  12nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171406(CHEMBL3804965)
Affinity DataEC50:  8.20nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171457(CHEMBL3805077)
Affinity DataEC50:  24nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171458(CHEMBL3806169)
Affinity DataEC50:  26nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171459(CHEMBL3805772)
Affinity DataEC50:  101nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171400(CHEMBL3805518)
Affinity DataEC50:  13nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171460(CHEMBL3805826)
Affinity DataEC50:  464nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171392(CHEMBL3805559)
Affinity DataEC50:  13nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171462(CHEMBL3805884)
Affinity DataEC50:  7.20nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171463(CHEMBL3806091)
Affinity DataEC50:  122nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171468(CHEMBL3804943)
Affinity DataEC50:  26nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171476(CHEMBL3806224)
Affinity DataEC50:  34nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171485(CHEMBL3806047)
Affinity DataEC50:  97nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171486(CHEMBL3805434)
Affinity DataEC50:  137nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171488(CHEMBL3805327)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171489(CHEMBL3805262)
Affinity DataEC50:  361nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171490(CHEMBL3805515)
Affinity DataEC50:  120nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171491(CHEMBL3805046)
Affinity DataEC50:  301nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171398(CHEMBL3804954)
Affinity DataEC50:  309nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171397(CHEMBL3805376)
Affinity DataEC50:  122nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171399(CHEMBL3805600)
Affinity DataEC50: >100nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataEC50:  285nMAssay Description:Agonistic activity at human 5-HT1A receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171405(CHEMBL3805165)
Affinity DataIC50: 4.10nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataIC50: 7nMAssay Description:Antagonistic activity at 5-HT2c receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171392(CHEMBL3805559)
Affinity DataIC50: 8.5nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171461(CHEMBL3805120)
Affinity DataIC50: 9.80nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171401(CHEMBL3805860)
Affinity DataIC50: 10nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataIC50: 10nMAssay Description:Antagonistic activity at alpha-1A adrenergic receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171402(CHEMBL3805099)
Affinity DataIC50: 12nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171468(CHEMBL3804943)
Affinity DataIC50: 12nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171400(CHEMBL3805518)
Affinity DataIC50: 15nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataIC50: 17nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171460(CHEMBL3805826)
Affinity DataIC50: 17nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171400(CHEMBL3805518)
Affinity DataIC50: 23nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171406(CHEMBL3804965)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171491(CHEMBL3805046)
Affinity DataIC50: 30nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171457(CHEMBL3805077)
Affinity DataIC50: 32nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171476(CHEMBL3806224)
Affinity DataIC50: 35nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171402(CHEMBL3805099)
Affinity DataIC50: 35nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171392(CHEMBL3805559)
Affinity DataIC50: 35nMAssay Description:Antagonistic activity at alpha-1A adrenergic receptor (unknown origin) after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171486(CHEMBL3805434)
Affinity DataIC50: 38nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171462(CHEMBL3805884)
Affinity DataIC50: 39nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171404(CHEMBL3805649)
Affinity DataIC50: 43nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171392(CHEMBL3805559)
Affinity DataIC50: 46nMAssay Description:Antagonistic activity at human 5-HT2A receptor assessed as calcium flux after 10 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Shanghai Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50171458(CHEMBL3806169)
Affinity DataIC50: 55nMAssay Description:Antagonistic activity at human dopamine D2 receptor measured after 60 mins by Ultra Lance cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2017
Entry Details Article
PubMed
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