Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50047441
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167961(CHEMBL3800596)
Affinity DataEC50:  121nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167960(CHEMBL3799512)
Affinity DataEC50:  15nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167959(CHEMBL3799242)
Affinity DataEC50:  65nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167929(CHEMBL3798702)
Affinity DataEC50:  38nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167928(CHEMBL3797699)
Affinity DataEC50:  770nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167927(CHEMBL3800090)
Affinity DataEC50:  60nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167926(CHEMBL3798871)
Affinity DataEC50:  234nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167925(CHEMBL3798047)
Affinity DataEC50:  37nMAssay Description:Inhibition of MetAP2 in HUVEC assessed as accumulation of N-Met-14-3-3gamma after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167916(CHEMBL3798615)
Affinity DataIC50: 3nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167926(CHEMBL3798871)
Affinity DataIC50: 4nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167915(CHEMBL3798727)
Affinity DataIC50: 4nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167929(CHEMBL3798702)
Affinity DataIC50: 5nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167960(CHEMBL3799512)
Affinity DataIC50: 5nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167959(CHEMBL3799242)
Affinity DataIC50: 5nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167922(CHEMBL3797286)
Affinity DataIC50: 5nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167961(CHEMBL3800596)
Affinity DataIC50: 6nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167917(CHEMBL3797663)
Affinity DataIC50: 6nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167919(CHEMBL3799449)
Affinity DataIC50: 8nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167920(CHEMBL3800546)
Affinity DataIC50: 8nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167921(CHEMBL3800534)
Affinity DataIC50: 8nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167918(CHEMBL3799467)
Affinity DataIC50: 9nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167923(CHEMBL3797707)
Affinity DataIC50: 10nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167914(CHEMBL3798034)
Affinity DataIC50: 11nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167927(CHEMBL3800090)
Affinity DataIC50: 11nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167925(CHEMBL3798047)
Affinity DataIC50: 13nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167924(CHEMBL3798381)
Affinity DataIC50: 15nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167909(CHEMBL3798509)
Affinity DataIC50: 20nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167928(CHEMBL3797699)
Affinity DataIC50: 21nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167922(CHEMBL3797286)
Affinity DataIC50: 50nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167910(CHEMBL3798100)
Affinity DataIC50: 62nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167904(CHEMBL3799496)
Affinity DataIC50: 79nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167913(CHEMBL3798443)
Affinity DataIC50: 91nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167923(CHEMBL3797707)
Affinity DataIC50: 100nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167920(CHEMBL3800546)
Affinity DataIC50: 200nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167907(CHEMBL3798111)
Affinity DataIC50: 220nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167915(CHEMBL3798727)
Affinity DataIC50: 316nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167916(CHEMBL3798615)
Affinity DataIC50: 316nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167912(CHEMBL3799532)
Affinity DataIC50: 360nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167917(CHEMBL3797663)
Affinity DataIC50: 398nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167918(CHEMBL3799467)
Affinity DataIC50: 501nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167919(CHEMBL3799449)
Affinity DataIC50: 501nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167911(CHEMBL3799684)
Affinity DataIC50: 550nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167908(CHEMBL3799625)
Affinity DataIC50: 730nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167906(CHEMBL3798664)
Affinity DataIC50: 960nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50209237(6-bromo-1H-indazole | CHEMBL247365)
Affinity DataIC50: 1.10E+3nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167914(CHEMBL3798034)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167901(CHEMBL3798369)
Affinity DataIC50: 2.80E+3nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetMicrotubule-associated protein 2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167905(CHEMBL3799845)
Affinity DataIC50: 5.50E+3nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167924(CHEMBL3798381)
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50167921(CHEMBL3800534)
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2017
Entry Details Article
PubMed
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