Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50047757
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187704(CHEMBL3828024)
Affinity DataIC50: 25nMAssay Description:Inhibition of PSMA (unknown origin) assessed as reduction in glutamate formation using NAAG as substrate preincubated for 30 mins followed by substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187705(CHEMBL3828668)
Affinity DataIC50: 28nMAssay Description:Inhibition of PSMA (unknown origin) assessed as reduction in glutamate formation using NAAG as substrate preincubated for 30 mins followed by substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50106240(6-Chloro-2-(2-hydroxy-biphenyl-3-yl)-1H-indole-5-c...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187705(CHEMBL3828668)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187711(CHEMBL3827463)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187707(CHEMBL3827292)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187708(CHEMBL3827374)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187709(CHEMBL3827645)
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187710(CHEMBL3827788)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187706(CHEMBL3828589)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187713(CHEMBL3828730)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50102768(2-(2-Hydroxy-phenyl)-1H-indole-5-carboxamidine | C...)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed
TargetSerine protease hepsin(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50187712(CHEMBL3828185)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of recombinant human hepsin using Boc-QAR-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details Article
PubMed