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Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50047405
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165203(CHEMBL3617113)
Affinity DataKi:  0.0430nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165207(CHEMBL1404528)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  0.850nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50024204(MESULERGINE | CHEMBL12314 | 4,7-dimethyl-(6aR,9S,1...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165203(CHEMBL3617113)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165320(CHEMBL3799165)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165212(CHEMBL3797981)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165210(CHEMBL3799209)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165209(CHEMBL3798450)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165208(CHEMBL3798863)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165207(CHEMBL1404528)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165206(CHEMBL3617211)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165205(CHEMBL3798961)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165204(CHEMBL3797474)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from 5HT2C receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165320(CHEMBL3799165)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165212(CHEMBL3797981)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165210(CHEMBL3799209)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165209(CHEMBL3798450)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165208(CHEMBL3798863)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165206(CHEMBL3617211)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165205(CHEMBL3798961)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50165204(CHEMBL3797474)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley rat brain cortex incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed