Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50001762
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017914(CHEMBL353950 | 3-(1-Ethyl-5-pyridin-3-ylmethyl-1H-...)
Affinity DataIC50: 42nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017903(CHEMBL170754 | 3-(1-tert-Butyl-5-pyridin-3-ylmethy...)
Affinity DataIC50: 44nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017905(CHEMBL352763 | 2-Methyl-3-(1-methyl-5-pyridin-3-yl...)
Affinity DataIC50: 50nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017909(CHEMBL170776 | 3-(5-Imidazol-1-ylmethyl-1-methyl-1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017896(CHEMBL11662 | (E)-3-(4-Imidazol-1-ylmethyl-phenyl)...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017912(CHEMBL169331 | 3-(5-Imidazol-1-ylmethyl-1-methyl-1...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017915(CHEMBL352512 | 3-(1-Isopropyl-5-pyridin-3-ylmethyl...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017908(CHEMBL167601 | 3-(5-Imidazol-1-ylmethyl-1-methyl-1...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017910(CHEMBL352874 | 3-(5-Imidazol-1-ylmethyl-1-methyl-1...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017901(CHEMBL169905 | 3-(5-Imidazol-1-ylmethyl-1H-pyrrol-...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017913(CHEMBL170615 | 2-(5-Imidazol-1-ylmethyl-1-methyl-1...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017898(CHEMBL354424 | 2-Methyl-3-(1-phenyl-5-pyridin-3-yl...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017907(CHEMBL262055 | 3-[1-(2,2-Dimethyl-propyl)-5-pyridi...)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed