Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50047268
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50156468(CHEMBL3792916)
Affinity DataIC50: 0.190nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 0.940nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161007(CHEMBL3792940)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50156470(CHEMBL3792842)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50156470(CHEMBL3792842)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161007(CHEMBL3792940)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161005(CHEMBL3793480)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161005(CHEMBL3793480)
Affinity DataIC50: 27nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161006(CHEMBL3794512)
Affinity DataIC50: 155nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50156468(CHEMBL3792916)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161004(CHEMBL3794076)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50156471(CHEMBL3793231)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50156471(CHEMBL3793231)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161006(CHEMBL3794512)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161003(CHEMBL3794468)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161004(CHEMBL3794076)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50161003(CHEMBL3794468)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MMP9 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed