Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50047375
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163389(CHEMBL3793278)
Affinity DataIC50: 220nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
LigandPNGBDBM50163389(CHEMBL3793278)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of KDM3C (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163393(CHEMBL3793435)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50343530(5,7-dichloro-4-((3-(4-methoxyphenylthio)benzyl)(me...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163387(CHEMBL3794377)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163392(CHEMBL1808018)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163390(CHEMBL3793690)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50320734(4-hydroxybenzohydrazide | 4-Hydroxy-benzoic acid h...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 4E(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163389(CHEMBL3793278)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of KDM4E (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163411(CHEMBL3793443)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50318639(6-hydroxy-1-methoxy-9H-xanthen-9-one | CHEMBL10842...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163430(CHEMBL3792463)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM34463(cid_848720 | SMR000077740 | 3-benzyl-6-(2-pyridiny...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 3A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163389(CHEMBL3793278)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of KDM3A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163388(CHEMBL3793686)
Affinity DataIC50: 6.40E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5A(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163436(CHEMBL3793454)
Affinity DataIC50: 8.30E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 6B(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163389(CHEMBL3793278)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of KDM6B (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50163389(CHEMBL3793278)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of KDM5B (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed