Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50047370
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50163307(CHEBI:66708 | 3,5-Dicaffeoylquinic Acid Methyl Est...)
Affinity DataIC50: 4.99E+3nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using fluor de lys as substrate after 10 to 15 mins by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM19410(benzamide-type inhibitor, 3 | CHEMBL27759 | pyridi...)
Affinity DataIC50: 6.73E+3nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using fluor de lys as substrate after 10 to 15 mins by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50163307(CHEBI:66708 | 3,5-Dicaffeoylquinic Acid Methyl Est...)
Affinity DataIC50: 7.59E+3nMAssay Description:Inhibition of HDAC in human HeLa cells using Boc-Lys(AC)-AMC as substrate after 24 to 48 hrs by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM19410(benzamide-type inhibitor, 3 | CHEMBL27759 | pyridi...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of HDAC in human HeLa cells using Boc-Lys(AC)-AMC as substrate after 24 to 48 hrs by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50362839(CHEMBL249447)
Affinity DataIC50: 1.43E+5nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using fluor de lys as substrate after 10 to 15 mins by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50163308(CHEBI:16384 | 3-O-Caffeoylquinic Acid | CHEMBL2494...)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using fluor de lys as substrate after 10 to 15 mins by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50327036(Chlorogenic acid (CGA) | (1R,3S,4S,5S)-3-[(E)-3-(3...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using fluor de lys as substrate after 10 to 15 mins by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50327036(Chlorogenic acid (CGA) | (1R,3S,4S,5S)-3-[(E)-3-(3...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HDAC in human HeLa cells using Boc-Lys(AC)-AMC as substrate after 24 to 48 hrs by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50163308(CHEBI:16384 | 3-O-Caffeoylquinic Acid | CHEMBL2494...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HDAC in human HeLa cells using Boc-Lys(AC)-AMC as substrate after 24 to 48 hrs by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50362839(CHEMBL249447)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of HDAC in human HeLa cells using Boc-Lys(AC)-AMC as substrate after 24 to 48 hrs by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed