Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50047368
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162967(CHEMBL3792850)
Affinity DataIC50: 9nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162967(CHEMBL3792850)
Affinity DataIC50: 10nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162968(CHEMBL3793843)
Affinity DataIC50: 23nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162968(CHEMBL3793843)
Affinity DataIC50: 34nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162971(CHEMBL3793804)
Affinity DataIC50: 42nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163005(CHEMBL3793847)
Affinity DataIC50: 43nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163003(CHEMBL3793427)
Affinity DataIC50: 46nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162970(CHEMBL3792973)
Affinity DataIC50: 56nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163011(CHEMBL3794211)
Affinity DataIC50: 61nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163007(CHEMBL3793695)
Affinity DataIC50: 90nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163009(CHEMBL3792878)
Affinity DataIC50: 95nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163030(CHEMBL3792955)
Affinity DataIC50: 107nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163032(CHEMBL3793933)
Affinity DataIC50: 110nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163022(CHEMBL3794503)
Affinity DataIC50: 113nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162967(CHEMBL3792850)
Affinity DataIC50: 137nMAssay Description:Inhibition of human N-terminal GST-tagged TRKA cytoplasmic domain (436 to 790 residues) expressed in baculovirus expression system using fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50163033(CHEMBL3794507)
Affinity DataIC50: 281nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162947(CHEMBL3794415)
Affinity DataIC50: 310nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM24634(N-phenyl-1H-indazole-3-carboxamide | indazole amid...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using fluorescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50331283(N-(4-methoxyphenyl)-1H-indazole-3-carboxamide | CH...)
Affinity DataIC50: 352nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162967(CHEMBL3792850)
Affinity DataIC50: 410nMAssay Description:Inhibition of human N-terminal GST-tagged HGK catalytic domain (1 to 328 residues) expressed in baculovirus expression system using fluorescence labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM24634(N-phenyl-1H-indazole-3-carboxamide | indazole amid...)
Affinity DataIC50: 417nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162948(CHEMBL3793590)
Affinity DataIC50: 443nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162942(CHEMBL3792695)
Affinity DataIC50: 552nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162945(CHEMBL3793337)
Affinity DataIC50: 786nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162969(CHEMBL3793334)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162966(CHEMBL3792787)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162951(CHEMBL3792750)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162950(CHEMBL3792669)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162949(CHEMBL3794143)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162946(CHEMBL3793040)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162944(CHEMBL3794579)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50162943(CHEMBL3792732)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptid...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2017
Entry Details Article
PubMed