Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50047470
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169211(CHEMBL3805284)
Affinity DataIC50: 11nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169216(CHEMBL3805336)
Affinity DataIC50: 20nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169093(CHEMBL3805908)
Affinity DataIC50: 60nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169094(CHEMBL3805524)
Affinity DataIC50: 69nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169219(CHEMBL3804890)
Affinity DataIC50: 84nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169161(CHEMBL3806139)
Affinity DataIC50: 94nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169174(CHEMBL3805345)
Affinity DataIC50: 101nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169208(CHEMBL3805800)
Affinity DataIC50: 222nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169172(CHEMBL3805882)
Affinity DataIC50: 232nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169133(CHEMBL3805506)
Affinity DataIC50: 308nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169223(CHEMBL3806295)
Affinity DataIC50: 325nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169205(CHEMBL3805131)
Affinity DataIC50: 491nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169092(CHEMBL3806080)
Affinity DataIC50: 716nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169097(CHEMBL3805947)
Affinity DataIC50: 746nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169186(CHEMBL3805174)
Affinity DataIC50: 763nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169120(CHEMBL3805758)
Affinity DataIC50: 917nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169123(CHEMBL3805419)
Affinity DataIC50: 937nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169154(CHEMBL3805399)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169163(CHEMBL3805823)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169139(CHEMBL3805511)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169177(CHEMBL3804961)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169091(CHEMBL3805909)
Affinity DataIC50: 3.27E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169117(CHEMBL3805968)
Affinity DataIC50: 3.37E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169220(CHEMBL3805066)
Affinity DataIC50: 3.83E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169131(CHEMBL3805815)
Affinity DataIC50: 8.96E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169119(CHEMBL3805334)
Affinity DataIC50: 9.68E+3nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169190(CHEMBL3805124)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169095(CHEMBL3804992)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169096(CHEMBL3805007)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169130(CHEMBL3805507)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169200(CHEMBL3805435)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169090(CHEMBL3805525)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169187(CHEMBL3804864)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169182(CHEMBL3805862)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169150(CHEMBL3805366)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetCholesteryl ester transfer protein(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169152(CHEMBL3805680)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CETP in 95% human serum assessed as suppression of transfer of [3H]-cholesterol oleate/[3H]-triolein from LDL to HDL after 1 hr by liqu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed