Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50010184
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University of Oklahoma Cobre In Structural Biology

Curated by ChEMBL
LigandPNGBDBM50535809(Sclerotiamide)
Affinity DataEC50:  3.96E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University of Oklahoma Cobre In Structural Biology

Curated by ChEMBL
LigandPNGBDBM50535810(CHEMBL4593796)
Affinity DataEC50:  2.22E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University of Oklahoma Cobre In Structural Biology

Curated by ChEMBL
LigandPNGBDBM50535809(Sclerotiamide)
Affinity DataEC50:  8.75E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University of Oklahoma Cobre In Structural Biology

Curated by ChEMBL
LigandPNGBDBM50535811(CHEMBL4549588)
Affinity DataEC50:  100nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University of Oklahoma Cobre In Structural Biology

Curated by ChEMBL
LigandPNGBDBM50535811(CHEMBL4549588)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using FITC-beta casein as substrate assessed as degradation of substrate peptide preincubated for 15 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetATP-dependent Clp protease proteolytic subunit(Escherichia coli (strain K12))
University of Oklahoma Cobre In Structural Biology

Curated by ChEMBL
LigandPNGBDBM50535810(CHEMBL4593796)
Affinity DataEC50:  2.54E+4nMAssay Description:Activation of Escherichia coli BLR (DE3) ClpP using Abz-DFAPKMALVPYNO2 as substrate assessed as degradation of substrate peptide preincubated for 15 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed