Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50006555
TargetTranscription factor 4(Human)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50436058(PNU-74654 | CHEMBL254381 | US9738628, Compound PNU...)
Affinity DataKd:  450nMAssay Description:Inhibition of His6 tagged Tcf4 1-53/beta catenin (unknown origin) interaction by VP-ITC titration calorimeter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTranscription factor 4(Human)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50500849(CHEMBL3780110)
Affinity DataIC50: 640nMAssay Description:Inhibition of human GST tagged Tcf4/beta catenin interaction after 2 hrs using fluorescent AP Attophos substrate by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTranscription factor 4(Human)
King Saud University

Curated by ChEMBL
LigandPNGBDBM32102(cid_66541 | 1,6-dimethylpyrimido[5,4-e][1,2,4]tria...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human GST tagged Tcf4/beta catenin interaction after 2 hrs using fluorescent AP Attophos substrate by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTranscription factor 4(Human)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50158807(3-butyryl-1,8-dihydroxy-2-methylphenanthrene-9,10-...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human GST tagged Tcf4/beta catenin interaction after 2 hrs using fluorescent AP Attophos substrate by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTranscription factor 4(Human)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50500850(CHEMBL261214)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human GST tagged Tcf4/beta catenin interaction after 2 hrs using fluorescent AP Attophos substrate by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTranscription factor 4(Human)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50500848(CHEMBL2397075)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human GST tagged Tcf4/beta catenin interaction after 2 hrs using fluorescent AP Attophos substrate by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCatenin beta-1/Transcription factor 4(Human)
King Saud University

Curated by ChEMBL
LigandPNGBDBM50500847(Cercosporin)
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of human GST tagged Tcf4/beta catenin interaction after 2 hrs using fluorescent AP Attophos substrate by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed