Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50047183
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152685(CHEMBL3780676)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152684(CHEMBL3781716)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152685(CHEMBL3780676)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of FLT3 (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152683(CHEMBL3781674)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152678(CHEMBL3780761)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152682(CHEMBL3780662)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152681(CHEMBL3781197)
Affinity DataIC50: 12nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152679(CHEMBL3780556)
Affinity DataIC50: 13nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152680(CHEMBL3780566)
Affinity DataIC50: 18nMAssay Description:Inhibition of cMet (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152685(CHEMBL3780676)
Affinity DataIC50: 363nMAssay Description:Inhibition of cKIT (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152685(CHEMBL3780676)
Affinity DataIC50: 527nMAssay Description:Inhibition of PDGFRbeta (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152685(CHEMBL3780676)
Affinity DataIC50: 543nMAssay Description:Inhibition of VEGFR-2 (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50152685(CHEMBL3780676)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed