Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50047282
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157303(CHEMBL3785774)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157313(CHEMBL3786892)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157313(CHEMBL3786892)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157538(CHEMBL3785299)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157538(CHEMBL3785299)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157534(CHEMBL3786402)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157303(CHEMBL3785774)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157534(CHEMBL3786402)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50436850(CHEMBL2403108 | CERITINIB | US10053458, Comparativ...)
Affinity DataIC50: 14nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157326(CHEMBL3785115)
Affinity DataIC50: 16nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157336(CHEMBL3785093)
Affinity DataIC50: 16nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157529(CHEMBL3786763)
Affinity DataIC50: 18nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157319(CHEMBL3786270)
Affinity DataIC50: 21nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157527(CHEMBL3785497)
Affinity DataIC50: 21nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157533(CHEMBL3786431)
Affinity DataIC50: 27nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50436850(CHEMBL2403108 | CERITINIB | US10053458, Comparativ...)
Affinity DataIC50: 29nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157528(CHEMBL3786127)
Affinity DataIC50: 29nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157318(CHEMBL3785322)
Affinity DataIC50: 34nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157529(CHEMBL3786763)
Affinity DataIC50: 37nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157530(CHEMBL3785538)
Affinity DataIC50: 40nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157527(CHEMBL3785497)
Affinity DataIC50: 40nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157530(CHEMBL3785538)
Affinity DataIC50: 40nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157528(CHEMBL3786127)
Affinity DataIC50: 42nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157317(CHEMBL3787539)
Affinity DataIC50: 43nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157344(CHEMBL3786792)
Affinity DataIC50: 44nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157323(CHEMBL3787262)
Affinity DataIC50: 52nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157319(CHEMBL3786270)
Affinity DataIC50: 56nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157533(CHEMBL3786431)
Affinity DataIC50: 94nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157326(CHEMBL3785115)
Affinity DataIC50: 97nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157336(CHEMBL3785093)
Affinity DataIC50: 100nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157318(CHEMBL3785322)
Affinity DataIC50: 109nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157346(CHEMBL3785384)
Affinity DataIC50: 122nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157344(CHEMBL3786792)
Affinity DataIC50: 200nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157323(CHEMBL3787262)
Affinity DataIC50: 201nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157317(CHEMBL3787539)
Affinity DataIC50: 207nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157351(CHEMBL3785480)
Affinity DataIC50: 212nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157346(CHEMBL3785384)
Affinity DataIC50: 222nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157316(CHEMBL3787367)
Affinity DataIC50: 342nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157322(CHEMBL3786831)
Affinity DataIC50: 424nMAssay Description:Inhibition of wild type ALK (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157322(CHEMBL3786831)
Affinity DataIC50: 600nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetALK tyrosine kinase receptor(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157316(CHEMBL3787367)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of ALK L1196M mutant (unknown origin) after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157303(CHEMBL3785774)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Chungbuk National University

Curated by ChEMBL
LigandPNGBDBM50157313(CHEMBL3786892)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed