Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50047583
TargetPotassium voltage-gated channel subfamily A member 3(Mouse)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50176999(CHEMBL3814333)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of mouse Kv1.3 expressed in L929 cells at -80 mV holding potential by whole cell patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 30nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 170nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/15/2017
Entry Details Article
PubMed