Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50047152
LigandPNGBDBM50151297(CHEMBL3771056)
Affinity DataIC50: 5nMAssay Description:Modulation of gamma-secretase activity (unknown origin) assessed as amyloid-beta(1-42) production by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50151298(CHEMBL3769869)
Affinity DataIC50: 21nMAssay Description:Modulation of gamma-secretase activity (unknown origin) assessed as amyloid-beta(1-42) production by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50151299(CHEMBL3770867)
Affinity DataIC50: 36nMAssay Description:Modulation of gamma-secretase activity (unknown origin) assessed as amyloid-beta(1-42) production by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed
TargetPresenilin-1(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50151300(CHEMBL3769891)
Affinity DataIC50: 56nMAssay Description:Modulation of gamma-secretase activity (unknown origin) assessed as amyloid-beta(1-42) production by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2017
Entry Details Article
PubMed