Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50047083
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147675(CHEMBL3764883)
Affinity DataIC50: 34nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147674(CHEMBL3763392)
Affinity DataIC50: 269nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147680(CHEMBL3763722)
Affinity DataIC50: 564nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147683(CHEMBL3765457)
Affinity DataIC50: 640nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 950nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147676(CHEMBL3763878)
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147677(CHEMBL3764880)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147684(CHEMBL3765105)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147684(CHEMBL3765105)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147685(CHEMBL3765574)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147688(CHEMBL3763205)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147681(CHEMBL3764119)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147685(CHEMBL3765574)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147676(CHEMBL3763878)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147681(CHEMBL3764119)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147685(CHEMBL3765574)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147683(CHEMBL3765457)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147679(CHEMBL3765110)
Affinity DataIC50: 5.77E+3nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147675(CHEMBL3764883)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147678(CHEMBL3763764)
Affinity DataIC50: 6.05E+3nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147674(CHEMBL3763392)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147681(CHEMBL3764119)
Affinity DataIC50: 7.12E+3nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147675(CHEMBL3764883)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147686(CHEMBL3763707)
Affinity DataIC50: 8.81E+3nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147688(CHEMBL3763205)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147685(CHEMBL3765574)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147684(CHEMBL3765105)
Affinity DataIC50: 9.94E+3nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147687(CHEMBL3765681)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147689(CHEMBL3763897)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147686(CHEMBL3763707)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147688(CHEMBL3763205)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147689(CHEMBL3763897)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147686(CHEMBL3763707)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147682(CHEMBL3765523)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kbeta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147678(CHEMBL3763764)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147676(CHEMBL3763878)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147689(CHEMBL3763897)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
LigandPNGBDBM50147674(CHEMBL3763392)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 60 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147677(CHEMBL3764880)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147688(CHEMBL3763205)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147683(CHEMBL3765457)
Affinity DataIC50: 2.03E+4nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147687(CHEMBL3765681)
Affinity DataIC50: 6.35E+4nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50147682(CHEMBL3765523)
Affinity DataIC50: 7.84E+4nMAssay Description:Inhibition of human DNA-PK using EPPLSQEAFADLWKK as substrate by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details Article
PubMed