Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50047222
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154931BDBM50154931(CHEMBL3775792)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50139171BDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154928BDBM50154928(CHEMBL3775509)
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154932BDBM50154932(CHEMBL3774632)
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154925BDBM50154925(CHEMBL3775470)
Affinity DataIC50: 8nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154930BDBM50154930(CHEMBL3774932)
Affinity DataIC50: 9nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154931BDBM50154931(CHEMBL3775792)
Affinity DataIC50: 9nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154929BDBM50154929(CHEMBL3775677)
Affinity DataIC50: 12nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 6309BDBM6309(8-cyclopentyl-6-acetyl-5-methyl-2-{[5-(piperazin-1...)
Affinity DataIC50: 16nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154923BDBM50154923(CHEMBL3775608)
Affinity DataIC50: 17nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154925BDBM50154925(CHEMBL3775470)
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154928BDBM50154928(CHEMBL3775509)
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154929BDBM50154929(CHEMBL3775677)
Affinity DataIC50: 21nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154932BDBM50154932(CHEMBL3774632)
Affinity DataIC50: 21nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154926BDBM50154926(CHEMBL3774979)
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154933BDBM50154933(CHEMBL3775502)
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154926BDBM50154926(CHEMBL3774979)
Affinity DataIC50: 37nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154924BDBM50154924(CHEMBL3775223)
Affinity DataIC50: 44nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50139171BDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 45nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154924BDBM50154924(CHEMBL3775223)
Affinity DataIC50: 46nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154935BDBM50154935(CHEMBL3775479)
Affinity DataIC50: 48nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154933BDBM50154933(CHEMBL3775502)
Affinity DataIC50: 49nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154922BDBM50154922(CHEMBL3774949)
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154923BDBM50154923(CHEMBL3775608)
Affinity DataIC50: 51nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154930BDBM50154930(CHEMBL3774932)
Affinity DataIC50: 54nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154927BDBM50154927(CHEMBL3775681)
Affinity DataIC50: 61nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154937BDBM50154937(CHEMBL518800)
Affinity DataIC50: 62nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154934BDBM50154934(CHEMBL3775606)
Affinity DataIC50: 70nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50139171BDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 72nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154920BDBM50154920(CHEMBL3774503)
Affinity DataIC50: 96nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154927BDBM50154927(CHEMBL3775681)
Affinity DataIC50: 114nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154922BDBM50154922(CHEMBL3774949)
Affinity DataIC50: 119nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50139171BDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 127nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154919BDBM50154919(CHEMBL3775467)
Affinity DataIC50: 132nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 7(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347389BDBM50347389(CHEMBL1801932)
Affinity DataIC50: 134nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 7533BDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 158nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154934BDBM50154934(CHEMBL3775606)
Affinity DataIC50: 165nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50139171BDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 178nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154920BDBM50154920(CHEMBL3774503)
Affinity DataIC50: 179nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154936BDBM50154936(CHEMBL3774434)
Affinity DataIC50: 183nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154936BDBM50154936(CHEMBL3774434)
Affinity DataIC50: 197nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154937BDBM50154937(CHEMBL518800)
Affinity DataIC50: 225nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154935BDBM50154935(CHEMBL3775479)
Affinity DataIC50: 229nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154932BDBM50154932(CHEMBL3774632)
Affinity DataIC50: 240nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154919BDBM50154919(CHEMBL3775467)
Affinity DataIC50: 422nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154921BDBM50154921(CHEMBL3775657)
Affinity DataIC50: 467nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50154932BDBM50154932(CHEMBL3774632)
Affinity DataIC50: 777nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 6309BDBM6309(8-cyclopentyl-6-acetyl-5-methyl-2-{[5-(piperazin-1...)
Affinity DataIC50: 892nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Palack£

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7533BDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of CDK5 (unknown origin) using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50154917BDBM50154917(CHEMBL3775861)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) expressed in sf9 cells using histone H1 as substrate in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
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