Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50006283
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498459(CHEMBL3596892)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498457(CHEMBL3596893)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498449(CHEMBL3596889)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498455(CHEMBL3596879)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498458(CHEMBL3596868)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498453(CHEMBL3596862)
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498449(CHEMBL3596889)
Affinity DataIC50: 56nMAssay Description:Inhibition of RET (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498459(CHEMBL3596892)
Affinity DataIC50: 63nMAssay Description:Inhibition of RET (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498457(CHEMBL3596893)
Affinity DataIC50: 64nMAssay Description:Inhibition of RET (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498452(CHEMBL3596873)
Affinity DataIC50: 92nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498458(CHEMBL3596868)
Affinity DataIC50: 120nMAssay Description:Inhibition of RET (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498453(CHEMBL3596862)
Affinity DataIC50: 140nMAssay Description:Inhibition of RET (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498452(CHEMBL3596873)
Affinity DataIC50: 210nMAssay Description:Inhibition of RET (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498455(CHEMBL3596879)
Affinity DataIC50: 330nMAssay Description:Inhibition of RET (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498460(CHEMBL3596858)
Affinity DataIC50: 380nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498462(CHEMBL3596870)
Affinity DataIC50: 420nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498456(CHEMBL3596874)
Affinity DataIC50: 490nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498454(CHEMBL3596876)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498450(CHEMBL3596864)
Affinity DataIC50: 870nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498455(CHEMBL3596879)
Affinity DataIC50: 880nMAssay Description:Inhibition of EphB2 (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498457(CHEMBL3596893)
Affinity DataIC50: 960nMAssay Description:Inhibition of KDR (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498459(CHEMBL3596892)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KDR (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498465(CHEMBL3596865)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498455(CHEMBL3596879)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of KDR (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498466(CHEMBL3596859)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498463(CHEMBL3596871)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498453(CHEMBL3596862)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of EphB2 (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498458(CHEMBL3596868)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of EphB2 (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498458(CHEMBL3596868)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of KDR (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498449(CHEMBL3596889)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of KDR (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498453(CHEMBL3596862)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of KDR (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498449(CHEMBL3596889)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of EphB2 (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498452(CHEMBL3596873)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of EphB2 (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498457(CHEMBL3596893)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of EphB2 (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498459(CHEMBL3596892)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of EphB2 (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498464(CHEMBL3596855)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498452(CHEMBL3596873)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of KDR (unknown origin) using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498461(CHEMBL3596856)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50498451(CHEMBL3596857)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant TrkA using ATP and 5FAM tagged TrkA peptide substrate incubated for 60 mins by microfluidics assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed