Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50047456
TargetMast/stem cell growth factor receptor Kit(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM77554(MLS001049144 | 7,8-dihydroxy-5,6-dimethoxy-2-pheny...)
Affinity DataIC50: 500nMAssay Description:Inhibition of N-terminal GST-His-tagged c-KIT (544 to 976 amino acids) D816V mutant (unknown origin) expressed in Sf9 insect cells using poly[Glu:Tyr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50064896(CHEMBL78010 | 5,7-dihydroxy-6-methoxy-2-(4-methoxy...)
Affinity DataIC50: 600nMAssay Description:Inhibition of N-terminal GST-His-tagged c-KIT (544 to 976 amino acids) D816V mutant (unknown origin) expressed in Sf9 insect cells using poly[Glu:Tyr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50079119(CHEMBL1171364)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of N-terminal GST-His-tagged c-KIT (544 to 976 amino acids) D816V mutant (unknown origin) expressed in Sf9 insect cells using poly[Glu:Tyr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50064896(CHEMBL78010 | 5,7-dihydroxy-6-methoxy-2-(4-methoxy...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of wild type His-tagged c-KIT (544 to 976 amino acids) (unknown origin) expressed in insect cells using poly[Glu:Tyr] (4:1) as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM77554(MLS001049144 | 7,8-dihydroxy-5,6-dimethoxy-2-pheny...)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of wild type His-tagged c-KIT (544 to 976 amino acids) (unknown origin) expressed in insect cells using poly[Glu:Tyr] (4:1) as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50079119(CHEMBL1171364)
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of wild type His-tagged c-KIT (544 to 976 amino acids) (unknown origin) expressed in insect cells using poly[Glu:Tyr] (4:1) as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50084980((2R,3R)-2-(3,4-dihydroxyphenyl)-3,4-dihydro-2H-chr...)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of N-terminal GST-His-tagged c-KIT (544 to 976 amino acids) D816V mutant (unknown origin) expressed in Sf9 insect cells using poly[Glu:Tyr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50084980((2R,3R)-2-(3,4-dihydroxyphenyl)-3,4-dihydro-2H-chr...)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of wild type His-tagged c-KIT (544 to 976 amino acids) (unknown origin) expressed in insect cells using poly[Glu:Tyr] (4:1) as substrate p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2017
Entry Details Article
PubMed