Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50047007
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143184(CHEMBL3759063)
Affinity DataIC50: 265nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase ATPase activity using pBR322 DNA as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143186(CHEMBL3759862)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase ATPase activity using pBR322 DNA as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143185(CHEMBL3759272)
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase ATPase activity using pBR322 DNA as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143184(CHEMBL3759063)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143185(CHEMBL3759272)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143186(CHEMBL3759862)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50449136(CHEMBL288959)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143189(CHEMBL3759276)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50414094(CHEMBL559696)
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143187(CHEMBL1481051)
Affinity DataIC50: 8.40E+5nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143188(CHEMBL1419183)
Affinity DataIC50: 8.40E+5nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMed
TargetDNA gyrase subunit B(Staphylococcus aureus)
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143190(CHEMBL3760057)
Affinity DataIC50: 8.40E+5nMAssay Description:Binding affinity to full length Staphylococcus aureus GyrB by STD-NMR spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/9/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)