Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50047000
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142919(CHEMBL3759860)
Affinity DataEC50:  46nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142926(CHEMBL3759759)
Affinity DataIC50: 52nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142909(CHEMBL3759928)
Affinity DataIC50: 66nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142929(CHEMBL3758309)
Affinity DataIC50: 68nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142928(CHEMBL3758976)
Affinity DataIC50: 73nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142921(CHEMBL3758433)
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142920(CHEMBL3759944)
Affinity DataEC50:  100nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50388686(CHEMBL74656)
Affinity DataEC50:  102nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142920(CHEMBL3759944)
Affinity DataIC50: 118nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142919(CHEMBL3759860)
Affinity DataIC50: 134nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142923(CHEMBL3758641)
Affinity DataIC50: 134nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142925(CHEMBL3758674)
Affinity DataIC50: 155nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142918(CHEMBL3759546)
Affinity DataIC50: 178nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142904(CHEMBL3759969)
Affinity DataIC50: 190nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142914(CHEMBL3758199)
Affinity DataEC50:  251nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142907(CHEMBL3759259)
Affinity DataIC50: 329nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142922(CHEMBL3758398)
Affinity DataIC50: 377nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142907(CHEMBL3759259)
Affinity DataEC50:  380nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50388686(CHEMBL74656)
Affinity DataIC50: 483nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142906(CHEMBL3759348)
Affinity DataIC50: 493nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142910(CHEMBL3758945)
Affinity DataIC50: 560nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142903(CHEMBL3759362)
Affinity DataIC50: 592nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142924(CHEMBL3758397)
Affinity DataIC50: 593nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142915(CHEMBL3758932)
Affinity DataIC50: 648nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142915(CHEMBL3758932)
Affinity DataEC50:  676nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142913(CHEMBL3759601)
Affinity DataEC50:  708nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142905(CHEMBL3759824)
Affinity DataIC50: 805nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142911(CHEMBL3758578)
Affinity DataIC50: 920nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142908(CHEMBL3758410)
Affinity DataIC50: 954nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142923(CHEMBL3758641)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50388686(CHEMBL74656)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142910(CHEMBL3758945)
Affinity DataEC50:  1.05E+3nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142912(CHEMBL3758523)
Affinity DataIC50: 1.12E+3nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142925(CHEMBL3758674)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142914(CHEMBL3758199)
Affinity DataIC50: 1.17E+3nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142913(CHEMBL3759601)
Affinity DataIC50: 1.27E+3nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142906(CHEMBL3759348)
Affinity DataEC50:  1.55E+3nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142924(CHEMBL3758397)
Affinity DataIC50: 2.86E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142909(CHEMBL3759928)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142922(CHEMBL3758398)
Affinity DataIC50: 4.58E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142917(CHEMBL3758721)
Affinity DataIC50: 5.76E+3nMAssay Description:Displacement of [3H]-GR113808 from human 5-HT4 receptor expressed in African green monkey COS7 cell membranes after 30 mins by liquid scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142909(CHEMBL3759928)
Affinity DataEC50:  6.03E+3nMAssay Description:Agonist activity at 5-HT4 receptor in rat esophageal thoracic muscularis mucosae assessed as carbachol-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142915(CHEMBL3758932)
Affinity DataIC50: 6.84E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142914(CHEMBL3758199)
Affinity DataIC50: 7.26E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142928(CHEMBL3758976)
Affinity DataIC50: 7.55E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142913(CHEMBL3759601)
Affinity DataIC50: 7.71E+3nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142905(CHEMBL3759824)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142904(CHEMBL3759969)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142926(CHEMBL3759759)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50142903(CHEMBL3759362)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG channel by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
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