Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50046929
TargetAcetylcholinesterase(Human)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of human acetylcholine esterase preincubated for 10 mins followed by the addition of 550 uM of acetylcholine iodide as substrate measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139052(CHEMBL3754700)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50: 5.65E+3nMAssay Description:Inhibition of human acetylcholine esterase preincubated for 10 mins followed by the addition of 550 uM of acetylcholine iodide as substrate measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139006(CHEMBL3753607)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139050(CHEMBL3753906)
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139051(CHEMBL3753070)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139006(CHEMBL3753607)
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139049(CHEMBL3753732)
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139007(CHEMBL3754287)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139052(CHEMBL3754700)
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139049(CHEMBL3753732)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139007(CHEMBL3754287)
Affinity DataIC50: 1.96E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase preincubated for 10 mins followed by the addition of acetylcholine iodide as substrate measured aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139050(CHEMBL3753906)
Affinity DataIC50: 2.28E+4nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139051(CHEMBL3753070)
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibition of horse butyrylcholine esterase preincubated for 10 mins followed by the addition of butyrylcholine iodide as substrate measured after 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139050(CHEMBL3753906)
Affinity DataKi:  8.60E+3nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139006(CHEMBL3753607)
Affinity DataKi:  1.04E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139052(CHEMBL3754700)
Affinity DataKi:  1.70E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139049(CHEMBL3753732)
Affinity DataKi:  1.90E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139051(CHEMBL3753070)
Affinity DataKi:  2.24E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139007(CHEMBL3754287)
Affinity DataKi:  2.24E+4nMAssay Description:Mixed inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
University of Bras£Lia

Curated by ChEMBL
LigandPNGBDBM50139053(CHEMBL3752227)
Affinity DataKi:  2.44E+4nMAssay Description:Non-competitive inhibition of electric eel acetylcholine esterase using acetylcholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed