Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50047114
TargetAmine oxidase [flavin-containing] A(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148940(CHEMBL3770019)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148936(CHEMBL3770489)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM39862(Selegiline | MLS000069378 | N-methyl-1-phenyl-N-pr...)
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148934(CHEMBL3770842)
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148937(CHEMBL3769637)
Affinity DataIC50: 68nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148941(CHEMBL3771328)
Affinity DataIC50: 204nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148933(CHEMBL3770005)
Affinity DataIC50: 218nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148939(CHEMBL3769586)
Affinity DataIC50: 523nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148935(CHEMBL3769956)
Affinity DataIC50: 627nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148938(CHEMBL3769915)
Affinity DataIC50: 2.46E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM15613(MCL | Aurorix | 4-chloro-N-[2-(morpholin-4-yl)ethy...)
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM29136(Iprazid | Euphozid | CHEMBL92401 | Iproniazid)
Affinity DataIC50: 6.56E+3nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM29136(Iprazid | Euphozid | CHEMBL92401 | Iproniazid)
Affinity DataIC50: 7.54E+3nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 6.14E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM39862(Selegiline | MLS000069378 | N-methyl-1-phenyl-N-pr...)
Affinity DataIC50: 6.73E+4nMAssay Description:Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50148932(CHEMBL3769733)
Affinity DataIC50: 6.94E+4nMAssay Description:Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI cells using p-tyramine as substrate after 15 mins by Amplex Red-based flu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2017
Entry Details Article
PubMed