Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50006469
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500099(CHEMBL3741765)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500092(CHEMBL3741937)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500097(CHEMBL3740962)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500105(CHEMBL3740249)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500103(CHEMBL3742211)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500098(CHEMBL3741101)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500106(CHEMBL3741673)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500094(CHEMBL3740203)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500101(CHEMBL1979298)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500091(CHEMBL3740563)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500100(CHEMBL3740034)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500095(CHEMBL2003928)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500107(CHEMBL3741464)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500102(CHEMBL3740606)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500109(CHEMBL3740547)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500093(CHEMBL2006267)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500096(CHEMBL3739720)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500108(CHEMBL3740917)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetCAAX prenyl protease 2(Human)
New York University Abu Dhabi

Curated by ChEMBL
LigandPNGBDBM50500104(CHEMBL3739592)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed