Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50001745
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  0.400nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50004823(CHEMBL298406 | Ecopipam | SCH 39166 | (6aS,13bR)-1...)
Affinity DataKi:  1.90nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017815(CHEMBL59139 | trans-11-Chloro-7-methyl-5,6a,7,8,9,...)
Affinity DataKi:  3.30nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017818(CHEMBL58205 | 7,11-Dimethyl-5,6a,7,8,9,13b-hexahyd...)
Affinity DataKi:  7.10nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017821(CHEMBL292451 | 12-Methoxy-7-methyl-5,6a,7,8,9,13b-...)
Affinity DataKi:  24nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017816(CHEMBL56100 | 7-Methyl-5,6a,7,8,9,13b-hexahydro-6H...)
Affinity DataKi:  68nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017820(CHEMBL294221 | 7-Methyl-5,6a,7,8,9,13b-hexahydro-6...)
Affinity DataKi:  73nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50010711(cis-(-) 11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahydr...)
Affinity DataKi:  474nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50010711(cis-(-) 11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahydr...)
Affinity DataKi:  513nMAssay Description:Inhibition of [3H]SCH-23390 binding to rat striatal homogenate dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50004823(CHEMBL298406 | Ecopipam | SCH 39166 | (6aS,13bR)-1...)
Affinity DataKi:  514nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50010715(CHEMBL58422 | (6aS,13bS)11-Chloro-7-methyl-5,6a,7,...)
Affinity DataKi:  531nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  648nMAssay Description:In vitro affinity of compound towards Dopamine receptor D2 was determined by measuring their ability to displace [3H]spiperone from rat striatal homo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50010712(CHEMBL294012 | (6aR,13bR)11-Chloro-7-methyl-5,6a,7...)
Affinity DataKi:  898nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017818(CHEMBL58205 | 7,11-Dimethyl-5,6a,7,8,9,13b-hexahyd...)
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017817(CHEMBL294215 | 12-Methoxy-7-methyl-5,6a,7,8,9,13b-...)
Affinity DataKi:  1.66E+3nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017819(CHEMBL301003 | 7-Methyl-5,6a,7,8,9,13b-hexahydro-6...)
Affinity DataKi:  1.73E+3nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017816(CHEMBL56100 | 7-Methyl-5,6a,7,8,9,13b-hexahydro-6H...)
Affinity DataKi:  2.41E+3nMAssay Description:In vitro affinity of compound towards Dopamine receptor D2 was determined by measuring their ability to displace [3H]spiperone from rat striatal homo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017821(CHEMBL292451 | 12-Methoxy-7-methyl-5,6a,7,8,9,13b-...)
Affinity DataKi:  2.48E+3nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50010715(CHEMBL58422 | (6aS,13bS)11-Chloro-7-methyl-5,6a,7,...)
Affinity DataKi:  3.05E+3nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017815(CHEMBL59139 | trans-11-Chloro-7-methyl-5,6a,7,8,9,...)
Affinity DataKi:  4.12E+3nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017823(CHEMBL294186 | 11-Methoxy-7-methyl-5,6a,7,8,9,13b-...)
Affinity DataKi:  4.20E+3nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017817(CHEMBL294215 | 12-Methoxy-7-methyl-5,6a,7,8,9,13b-...)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017820(CHEMBL294221 | 7-Methyl-5,6a,7,8,9,13b-hexahydro-6...)
Affinity DataKi:  7.87E+3nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50010711(cis-(-) 11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahydr...)
Affinity DataKi:  9.07E+3nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50010711(cis-(-) 11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahydr...)
Affinity DataKi:  9.07E+3nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50010712(CHEMBL294012 | (6aR,13bR)11-Chloro-7-methyl-5,6a,7...)
Affinity DataKi:  1.63E+4nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017822(CHEMBL442740 | 12-Methoxy-7-methyl-5,6a,7,8,9,13b-...)
Affinity DataKi:  2.44E+4nMAssay Description:In vitro affinity of compound towards dopamine (D1) receptor was determined by measuring their ability to displace [3H]SCH-23,390 from rat striatal h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017822(CHEMBL442740 | 12-Methoxy-7-methyl-5,6a,7,8,9,13b-...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017819(CHEMBL301003 | 7-Methyl-5,6a,7,8,9,13b-hexahydro-6...)
Affinity DataKi: >1.00E+5nMAssay Description:In vitro affinity of compound towards Dopamine receptor D2 was determined by measuring their ability to displace [3H]spiperone from rat striatal homo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM50017823(CHEMBL294186 | 11-Methoxy-7-methyl-5,6a,7,8,9,13b-...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]spiperone from rat striatal homogenate dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed