Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50046936
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142189(US9487512, 5 | CHEMBL3759239 | US10329256, Example...)
Affinity DataIC50: 62nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142076(CHEMBL3758988)
Affinity DataIC50: 77nMAssay Description:Covalent inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataIC50: 78nMAssay Description:Inhibition of rat MAO-B using benzylamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataIC50: 290nMAssay Description:Inhibition of rat MAO-A using serotonin as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142189(US9487512, 5 | CHEMBL3759239 | US10329256, Example...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant human MAO-B after 60 mins MAO-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142189(US9487512, 5 | CHEMBL3759239 | US10329256, Example...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant human MAO-A after 60 mins MAO-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50236898((1S,2R)-(+)-2-phenylcyclopropylamine | trans-2-phe...)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of LSD1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142238(CHEMBL3759201)
Affinity DataIC50: 8.76E+4nMAssay Description:Inhibition of recombinant human AKT for 60 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142238(CHEMBL3759201)
Affinity DataKi:  29nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142187(CHEMBL3758634)
Affinity DataKi:  46nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142237(CHEMBL3759797)
Affinity DataKi:  58nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142242(CHEMBL3759102)
Affinity DataKi:  88nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50139118(CHEMBL3759351)
Affinity DataKi:  150nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142240(CHEMBL3759861)
Affinity DataKi:  200nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50139119(CHEMBL3758849)
Affinity DataKi:  220nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142249(CHEMBL3759939)
Affinity DataKi:  220nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142079(CHEMBL3758636)
Affinity DataKi:  380nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142086(CHEMBL3758396)
Affinity DataKi:  540nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142235(CHEMBL3758821)
Affinity DataKi:  570nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142243(CHEMBL3758340)
Affinity DataKi:  650nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142185(CHEMBL3759654)
Affinity DataKi:  740nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142239(CHEMBL3760120)
Affinity DataKi:  800nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142236(CHEMBL3760085)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142186(CHEMBL3760091)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142077(CHEMBL3759070)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142080(CHEMBL3758211)
Affinity DataKi:  1.80E+3nMAssay Description:Competitive inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using 2 to 100 uM dimethylated H3K4 peptide substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142080(CHEMBL3758211)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50140245(CHEMBL3759574)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142187(CHEMBL3758634)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of recombinant human MAO-B after 60 mins MAO-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142075(CHEMBL3758747)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142248(CHEMBL3759283)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142241(CHEMBL3759645)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142188(CHEMBL3759472)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50139120(CHEMBL3759088)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142084(CHEMBL3758284)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142237(CHEMBL3759797)
Affinity DataKi:  9.70E+3nMAssay Description:Inhibition of recombinant human MAO-B after 60 mins MAO-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142080(CHEMBL3758211)
Affinity DataKi:  1.06E+4nMAssay Description:Inhibition of recombinant human MAO-B after 60 mins MAO-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142245(CHEMBL3758933)
Affinity DataKi:  1.65E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142238(CHEMBL3759201)
Affinity DataKi:  1.87E+4nMAssay Description:Inhibition of recombinant human MAO-B after 60 mins MAO-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142234(CHEMBL3758402)
Affinity DataKi:  2.23E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142083(CHEMBL3758664)
Affinity DataKi:  2.62E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142082(CHEMBL3758833)
Affinity DataKi:  3.22E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50139121(CHEMBL3759462)
Affinity DataKi:  4.38E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142078(CHEMBL3759840)
Affinity DataKi:  4.78E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142195(CHEMBL3759525)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142247(CHEMBL3759745)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142194(CHEMBL3758505)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetLysine-specific histone demethylase 1A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50139122(CHEMBL3758241)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged LSD1 catalytic domain (172 to 833 residues) using dimethylated H3K4 peptide substrate preincubated for 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142237(CHEMBL3759797)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human MAO-A after 60 mins MAO-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50142238(CHEMBL3759201)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human MAO-A after 60 mins MAO-glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2017
Entry Details Article
PubMed
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